Id: acc2517
Group: 1sens
Protein: stathmin
Gene Symbol: STMN1
Protein Id: P16949
Protein Name: STMN1_HUMAN
PTM: phosphorylation
Site: Ser38
Site Sequence: KESVPEFPLSPPKKKDLSLEE
Disease Category: Cancer
Disease: Ovarian Cancer
Disease Subtype: clear cell carcinoma
Disease Cellline: RMG-1
Disease Info:
Drug: paclitaxel
Drug Info: "Paclitaxel is a plant-derived alkaloid and potent antineoplastic agent that stabilizes microtubules to inhibit cancer cell division, primarily used in the treatment of ovarian, breast, and lung cancers. "
Effect: reduce
Effect Info: "Eribulin-induced stathmin phosphorylation is partially mediated by PP2A downregulation, which reduces the activity of stathmin and enhances the antiproliferative effect of paclitaxel on ovarian cancer."
Note: site unclear
Score: 5.0
Pubmed(PMID): 36328498
Sentence Index:
Sentence:

Sequence & Structure:

MASSDIQVKELEKRASGQAFELILSPRSKESVPEFPLSPPKKKDLSLEEIQKKLEAAEERRKSHEAEVLKQLAEKREHEKEVLQKAIEENNNFSKMAEEKLTHKMEANKENREAQMAAKLERLREKDKHIEEVRKNKESKDPADETEAD

No data.

Known Drugs:

source: Multi-Sources

(see table)

No data.

Protein Tractability:

source: Open Targets
Small molecule
Antibody
PROTAC
Other modalities
Approved Drug
Advanced Clinical
Phase 1 Clinical
Structure with Ligand
High-Quality Ligand
High-Quality Pocket
Med-Quality Pocket
Druggable Family
Approved Drug
Advanced Clinical
Phase 1 Clinical
UniProt loc high conf
GO CC high conf
UniProt loc med conf
UniProt SigP or TMHMM
GO CC med conf
Human Protein Atlas loc
Approved Drug
Advanced Clinical
Phase 1 Clinical
Literature
UniProt Ubiquitination
Database Ubiquitination
Half-life Data
Small Molecule Binder
Approved Drug
Advanced Clinical
Phase 1 Clinical

PTM Intensity:

source: CPTAC
STMN1-Ser38
Cancer Intensity
BRCA -1.168
COAD 1.155
HGSC -0.587
ccRCC 0.172
GBM -1.894
HNSC 0.771
LUAD 0.51
LUSC 0.588
non_ccRCC -1.017
PDAC 0.853
UCEC 0.617

PTM-Disease Association:

source: PTMD
Residue Position State Disease Class PMID
S 38 D Fanconi anemia Phosphorylation 26466335
S 38 D Alzheimer's disease Phosphorylation 16925597
S 38 P Endometrial cancer/carcinoma Phosphorylation 23538402
S 38 U Breast cancer Phosphorylation 26087399 27130664
S 38 U Schizophrenia Phosphorylation 16925597

State Note: Based on the distinct PTM states in diseases, PTMD classified all disease-associated PTMs into six classes, including whether the up-regulation (U) or down-regulation (D) of PTM levels, the absence (A) or presence (P) of PTMs, and the creation (C) or disruption (N) of PTM sites are associated with diseases.

PTM-Drug Perturbation Response:

source: DecryptM
Protein Gene PTM Position Modified sequence Cell Drug pEC50 Regulation Experiment
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 8.3711 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 8.267 up
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.5742 up
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.5609 up
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 6.9543 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 7.4166 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 7.257 up
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 8.6677 up
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.9297 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 7.7605 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 7.7221 up
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 6.9176 up
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 6.1302 up
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -3.0295 up
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK A431 Afatinib 8.5847 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Staursporin 6.2619 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Staursporin 6.2115 down
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Staursporin 6.1754 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK BT-474 Lapatinib 6.9895 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK BT-474 Lapatinib 6.8899 down
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK HeLa CUDC101 4.3434 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK PC-9 Lapatinib 4.69 down
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 8.1883 down
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 7.6554 down
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.6547 down
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Afatinib 8.7353 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Afatinib 8.2921 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A431 Afatinib 6.7609 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Afatinib 9.0483 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK A431 Afatinib 8.9141 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Afatinib 5.4488 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A431 Afatinib 2 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Afatinib 8.9405 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Afatinib 6.2203 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Afatinib 7.8143 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Afatinib 7.5188 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Dasatinib 11.7841 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Dasatinib 10.4952 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A431 Dasatinib 9.4703 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A431 Dasatinib 8.9977 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Dasatinib 8.9186 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A431 Dasatinib 8.8578 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Dasatinib 6.5808 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A431 Dasatinib 9.9492 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Dasatinib 9.9403 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Dasatinib 9.926 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK A431 Dasatinib 5.4336 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Dasatinib 10.0213 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Dasatinib 7.242 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Dasatinib 10.2396 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Dasatinib 8.5058 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Gefitinib 7.265 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Gefitinib 6.7746 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Gefitinib 9.9943 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Gefitinib 8.0103 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A431 Gefitinib 8.703 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Gefitinib 8.4461 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Gefitinib 8.0046 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK A431 Gefitinib 6.2624 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Gefitinib 13.9591 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Gefitinib 7.1704 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A431 Imatinib 9.425 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A431 Imatinib 8.9912 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A431 Imatinib 2 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 AZD8055 10.7135 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 AZD8055 10.5831 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 AZD8055 9.8617 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 AZD8055 7.2917 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 AZD8055 5.1808 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 Dactolisib 15 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Dactolisib 7.2704 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Dactolisib 6.2619 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Dactolisib 6.0781 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Dactolisib 5.8436 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Dactolisib 2 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Dasatinib 10.6043 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Dasatinib 8.9728 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Dasatinib 8.3916 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Dasatinib 8.2435 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Dasatinib 7.0189 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Dasatinib 5.6202 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Dasatinib 4.2844 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Dasatinib 2 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 MK2206 10.9144 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 MK2206 9.4462 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 MK2206 7.0347 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 MK2206 6.4952 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 MK2206 6.3508 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Nintedanib 11.0402 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 Nintedanib 8.9463 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Nintedanib 8.8456 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Nintedanib 8.7654 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Nintedanib 6.7715 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Nintedanib 6.5303 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 PD325901 15 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 PD325901 11.0136 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 PD325901 10.7361 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 PD325901 9.1645 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 PD325901 8.9997 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 PD325901 7.8696 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 PD325901 7.3983 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 PD325901 4.4803 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 Pictilisib 11.1523 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Pictilisib 10.8876 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Pictilisib 8.7561 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Pictilisib 8.2404 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Pictilisib 7.8744 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Pictilisib 7.367 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Refametinib 9.571 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Refametinib 8.765 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Refametinib 8.7163 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Refametinib 8.262 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Refametinib 2 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 Staursporin 6.1858 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Staursporin 6.0189 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK A549 Tideglusib 10.7988 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK A549 Tideglusib 9.0165 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK A549 Tideglusib 8.8047 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK A549 Tideglusib 8.3156 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK A549 Tideglusib 5.3595 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK A549 Tideglusib 2 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab 1.3802 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab 1.1838 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK ARH-77 Rituximab 0.0537 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK ARH-77 Rituximab -0.2383 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab -1.2202 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab -1.2203 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab -4.1423 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab 0.9448 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab -0.03 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab -0.081 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab -1.2169 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab -1.2187 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab -4.2544 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab -1.2035 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK ARH-77 Rituximab -1.2196 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab -3.7767 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab -3.8465 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab -3.9751 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK ARH-77 Rituximab -3.9841 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab -4.0555 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab -4.1854 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab 2.2839 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab 0.852 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab 0.0668 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK ARH-77 Rituximab 2.2173 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK ARH-77 Rituximab 1.6571 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK ARH-77 Rituximab -4.4778 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK BT-474 Lapatinib 4.4316 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK BT-474 Pertuzumab -1.9698 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK BT-474 Pertuzumab -2.9853 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK BT-474 Pertuzumab -4.2449 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK BT-474 Pertuzumab -4.3264 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK BT-474 Pertuzumab -6.0267 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK BT-474 Trastuzumab -2.569 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK BT-474 Trastuzumab -2.71 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK HeLa A485 10.8164 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK HeLa A485 10.4729 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa A485 10.2088 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK HeLa A485 6.2301 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK HeLa A485 5.2664 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK HeLa A486 14 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK HeLa A486 14 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa A486 11.1116 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK HeLa A486 5.2393 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK HeLa CUDC101 13.5229 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK HeLa CUDC101 7.187 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa CUDC101 5.2696 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK HeLa CUDC101 4.6943 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK HeLa Curcumin 9.5712 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK HeLa Curcumin 7.4504 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa Curcumin 5.5379 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK HeLa Curcumin 5.4809 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa Romidepsin 8.4875 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK HeLa Romidepsin 8.3082 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK HeLa SAHA 5.7602 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK HeLa SAHA 2.4332 -
P16949 STMN1 P Ser28;Ser38 S(ph)KESVPEFPLS(ph)PPK K562 Dasatinib 9.3588 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 9.2579 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK K562 Dasatinib 9.2564 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 9.2492 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 9.2441 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 9.239 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.2186 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 9.134 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.123 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 8.2172 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK K562 Dasatinib 8.0024 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 7.8319 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 7.7709 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 7.2622 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK K562 Dasatinib 6.2727 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 6.2586 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK K562 Dasatinib 11.0187 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 10.7753 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 10.6265 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 9.3226 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.2862 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 9.2821 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.2784 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 9.2644 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 7.7298 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.7585 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 9.736 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK K562 Dasatinib 9.6547 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Dasatinib 9.5178 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Dasatinib 9.3206 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 9.2649 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Dasatinib 8.9686 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Dasatinib 8.9112 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK K562 Imatinib 14.2627 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK K562 Imatinib 11.0646 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK K562 Imatinib 8.2464 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK K562 Imatinib 7.2624 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK K562 Imatinib 7.0553 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK K562 Imatinib 6.9948 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK KYSE-520 SHP099 8.3986 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK KYSE-520 SHP099 7.0624 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK KYSE-520 SHP099 6.2517 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK KYSE-520 SHP099 6.2494 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK KYSE-520 SHP099 5.4444 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK KYSE-520 SHP099 5.4019 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK KYSE-520 SHP099 5.2785 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK MDA-MB-175 Lapatinib 10.0044 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK MDA-MB-175 Lapatinib 7.535 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK MDA-MB-175 Lapatinib 7.175 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK MDA-MB-175 Pertuzumab -1.2201 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK MDA-MB-175 Pertuzumab -2.2044 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK MDA-MB-175 Trastuzumab 2.1007 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK MDA-MB-175 Trastuzumab -2.7378 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK MDA-MB-175 Trastuzumab -3.0369 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK PC-9 AZD4547 6.973 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK PC-9 AZD4547 5.265 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK PC-9 AZD4547 5.2589 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK PC-9 AZD4547 5.2551 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK PC-9 Lapatinib 7.2417 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK PC-9 Lapatinib 5.973 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK PC-9 Lapatinib 4.7594 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK PC-9 Lapatinib 4.6981 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK PC-9 LapatinibAZD4547 6.7369 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK PC-9 LapatinibAZD4547 6.6114 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK PC-9 LapatinibAZD4547 5.3551 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK PC-9 LapatinibAZD4547 5.2703 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK PC-9 LapatinibAZD4547 5.242 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK Ramos Rituximab 5.5229 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK Ramos Rituximab 1.7674 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK Ramos Rituximab -0.9843 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -1.2958 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab -2.8773 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab 2.3156 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK Ramos Rituximab -1.9534 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK Ramos Rituximab -2.4784 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK Ramos Rituximab -2.7321 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK Ramos Rituximab -3.199 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -3.4239 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab -1.3745 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK Ramos Rituximab -2.7069 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK Ramos Rituximab -2.7267 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -2.7279 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK Ramos Rituximab -4.2495 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab -2.82 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -2.8235 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK Ramos Rituximab -2.8432 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK Ramos Rituximab -2.9087 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab -0.8097 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -0.9807 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK Ramos Rituximab -2.1954 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK Ramos Rituximab -2.237 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK Ramos Rituximab -2.2391 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK Ramos Rituximab -1.7345 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK Ramos Rituximab -1.7844 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK Ramos Rituximab -2.2799 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK Ramos Rituximab -4.2398 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 9.4811 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 8.1033 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.5209 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.1924 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 6.6348 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 6.5235 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 16 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 12.36 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 12.1683 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 11.9207 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 9.7863 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 9.7503 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.9091 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 7.6219 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 7.4937 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.4627 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 6.5745 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 3 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 16 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 12.3619 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 12.1907 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 12.1475 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 10.4616 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 10.1623 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 9.1179 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 8.7524 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 8.6179 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 8.4449 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.1478 -
P16949 STMN1 P Ser31;Ser38 SKES(ph)VPEFPLS(ph)PPK RPMI8226 BTZ 6.4444 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 12.5919 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 12.5554 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 11.8583 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 10.1822 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.6687 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.4415 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 7.3839 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 7.3576 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 7.2571 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK RPMI8226 BTZ 6.426 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK RPMI8226 BTZ 3.9496 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 3.0167 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 16 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 8.8662 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK RPMI8226 BTZ 8.727 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.655 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.4412 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 7.4028 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK RPMI8226 BTZ 7.3445 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK RPMI8226 BTZ 4.365 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SK-BR-3 Lapatinib 7.8497 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SK-BR-3 Lapatinib 7.2624 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SK-BR-3 Lapatinib 7.22 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SK-BR-3 Pertuzumab 3.9073 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SK-BR-3 Pertuzumab 2.1465 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SK-BR-3 Pertuzumab -3.1333 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SK-BR-3 Trastuzumab 2.7008 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKKK SK-BR-3 Trastuzumab -2.2017 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SK-BR-3 Trastuzumab -2.2095 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SK-BR-3 Trastuzumab -2.763 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.2772 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.3286 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.5016 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.2707 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SU-DHL-4 Rituximab -1.2807 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.3 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -3.0081 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SU-DHL-4 Rituximab 1.0302 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.5192 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -2.9389 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -4.2381 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -3.2268 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SU-DHL-4 Rituximab -1.4405 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -3.2574 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -3.5813 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab 1.9546 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.4519 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.4525 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.5877 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.3791 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPKKK SU-DHL-4 Rituximab -1.4041 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.4264 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.4383 -
P16949 STMN1 P Ser38 SKESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.1344 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPKK SU-DHL-4 Rituximab -1.1648 -
P16949 STMN1 P Ser38 ESVPEFPLS(ph)PPK SU-DHL-4 Rituximab -1.2242 -

pEC50 Note: pEC50 is the negative logarithm of EC50 (half-maximal effective concentration, dosage unit Mol), calculated as pEC50 = -log10(EC50), which quantifies the potency of a drug or compound.

Function score:

source: funscoR

No data.

Cross Links: