Id: | acc4095 |
Group: | 1sens |
Protein: | CREB |
Gene Symbol: | Creb1 |
Protein Id: | P15337 |
Protein Name: | CREB1_RAT |
PTM: | phosphorylation |
Site: | Ser133 |
Site Sequence: | LNDLSSDAPGVPRIEEEKSEE |
Disease Category: | Cardiovascular and circulatory system diseases |
Disease: | Infarction |
Disease Subtype: | |
Disease Cellline: | |
Disease Info: | |
Drug: | Tat-NR2B9c |
Drug Info: | Tat - NR2B9c is a drug that may have potential effects in relevant medical fields. Its specific functions and applications may require further research and exploration. |
Effect: | modulate |
Effect Info: | "In the cerebral ischemia model, Tat-NR2B9c can selectively and persistently enhance the phosphorylation level of CaMKIV, thereby significantly reducing the volume of cerebral infarction and exhibiting neuroprotective effects." |
Note: | |
Score: | 4.0 |
Pubmed(PMID): | 23363435 |
Sentence Index: | 23363435_7 |
Sentence: | Tat-NR2B9c application significantly reduces infarct size and causes a selective and sustained elevation in CaMKIV phosphorylationation; effects which are blocked by coadministration of KN93. |
Sequence & Structure:
MTMDSGADNQQSGDAAVTEAESQQMTVQAQPQIATLAQVSMPAAHATSSAPTVTLVQLPNGQTVQVHGVIQAAQPSVIQSPQVQTVQISTIAESEDSQESVDSVTDSQKRREILSRRPSYRKILNDLSSDAPGVPRIEEEKSEEETSAPAITTVTVPTPIYQTSSGQYIAITQGGAIQLANNGTDGVQGLQTLTMTNAAATQPGTTILQYAQTTDGQQILVPSNQVVVQAASGDVQTYQIRTAPTSTIAPGVVMASSPALPTQPAEEAARKREVRLMKNREAARECRRKKKEYVKCLENRVAVLENQNKTLIEELKALKDLYCHKSD
Select PDB:
No data.
Protein Tractability:
source: Open TargetsNo data.
PTM Intensity:
source: CPTACNo data.
PTM-Disease Association:
source: PTMDResidue | Position | State | Disease | Class | PMID |
---|---|---|---|---|---|
S | 133 | U | Pulmonary hypertension | Phosphorylation | 34635097 |
State Note: Based on the distinct PTM states in diseases, PTMD classified all disease-associated PTMs into six classes, including whether the up-regulation (U) or down-regulation (D) of PTM levels, the absence (A) or presence (P) of PTMs, and the creation (C) or disruption (N) of PTM sites are associated with diseases.
PTM-Drug Perturbation Response:
source: DecryptMNo data.
Function score:
source: funscoRNo data.