Id: acc4867
Group: 1sens
Protein: p70S6K
Gene Symbol: Rps6kb1
Protein Id: P67999
Protein Name: KS6B1_RAT
PTM: phosphorylation
Site: Ser389
Site Sequence: SQFDSKFTRQTPVDSPDDSTL
Disease Category: Cardiovascular and circulatory system diseases
Disease: Cardiac Hypertrophy
Disease Subtype:
Disease Cellline: NNVMs
Disease Info:
Drug: Rapamycin
Drug Info: Rapamycin is a macrolide compound that is used as an immunosuppressant and has potential applications in treating various diseases such as cancer and aging-related conditions.
Effect: modulate
Effect Info: Rapamycin exerts its anti - hypertrophic effect by inhibiting the phosphorylation of p70S6K and regulating the expression of SUR2A protein.
Note:
Score: 4.0
Pubmed(PMID): 36988388
Sentence Index:
Sentence:

Sequence & Structure:

MRRRRRRDGFYPAPDFRHREAEDMAGVFDIDLDQPEDAGSEDELEEGGQLNESMDHGGVGPYELGMEHCEKFEISETSVNRGPEKIRPECFELLRVLGKGGYGKVFQVRKVTGANTGKIFAMKVLKKAMIVRNAKDTAHTKAERNILEEVKHPFIVDLIYAFQTGGKLYLILEYLSGGELFMQLEREGIFMEDTACFYLAEISMALGHLHQKGIIYRDLKPENIMLNHQGHVKLTDFGLCKESIHDGTVTHTFCGTIEYMAPEILMRSGHNRAVDWWSLGALMYDMLTGAPPFTGENRKKTIDKILKCKLNLPPYLTQEARDLLKKLLKRNAASRLGAGPGDAGEVQAHPFFRHINWEELLARKVEPPFKPLLQSEEDVSQFDSKFTRQTPVDSPDDSTLSESANQVFLGFTYVAPSVLESVKEKFSFEPKIRSPRRFIGSPRTPVSPVKFSPGDFWGRGASASTANPQTPVEYPMETSGIEQMDVTTSGEASAPLPIRQPNSGPYKKQAFPMISKRPEHLRMNL

No data.

Known Drugs:

source: Multi-Sources

(see table)

No data.

Protein Tractability:

source: Open Targets

No data.

PTM Intensity:

source: CPTAC

No data.

PTM-Disease Association:

source: PTMD

No data.

PTM-Drug Perturbation Response:

source: DecryptM

No data.

Function score:

source: funscoR

No data.

Cross Links: